Table of Compounds



1592U89

(1S,4R)-4-[2-amino-6-cyclopropyl-amino)-9H-purin-9-yl]-2-cyclopentene-1-methanol succinate (a carbovir analogue, Glaxo Wellcome)

3TC

(-)-b-L-2',3'-dideoxy-3'-thiacytidine (Glaxo Wellcome)

1737

Tetrahydronapthalene lignan derivative

a-APA R18893

a-nitro-anilino-phenylacetamide

A-77003, A-75925, A-80987

C2 symmetry-based protease inhibitors (Abbott Laboratories)

AAP-BHAP

bisheteroarylpiperazine analogue (Pharmacia & Upjohn)

ABT-378

Protease inhibitor

ABT-538

C2 symmetry-based protease inhibitor (Abbott Laboratories)

ADAMII

Methyl 3',3''-dichloro-4',4''-dimethoxy-5',5''-bis(methoxycarbonyl)-6,6-diphenyl-5-hexenoate. An alkenyldiarylmethane

AZdU

3'-azido-2',3'-dideoxyuridine

AZT

3'-azido-3'-deoxythymidine (Glaxo Wellcome)

AZT-p-ddI

3'-azido-3'-deoxythymidilyl-(5',5')-2',3'-dideoxyinosinic acid (Ivax)

BHAP

bisheteroarylpiperazine

BILA 1906

N-{1S-[[[3-[2S-(1,1-dimethylethyl)amino]carbonyl}-4R-]3-pyridinylmethyl)thio]-1-piperidinyl]-2R-hydroxy-1S-(phenylmethyl)propyl]amino]carbonyl]-2-methylpropyl}-2-quinolinecarboxamide (Bio-Mega/Boehringer Ingelheim)

BILA 2185

N-(1,1-dimethylethyl)-1-[2S-[[2-2,6-dimethyphenoxy)-1-oxoethyl]amino]-2R-hydroxy-4-phenylbutyl]4R-pyridinylthio)-2-piperidine-carboxamide (Bio-Mega/Boehringer Ingelheim)

BM+51.0836

thiazolo-isoindolinone derivative

BMS 186,318

aminodiol derivative HIV-1 protease inhibitor (Bristol-Myers Squibb)

d4API

9-[2,5-dihydro-5-(phosphonomethoxy)-2-furanel]adenine (Gilead Sciences)

d4C

2',3'-didehydro-2',3'-dideoxycytidine

d4T

2',3'-didehydro-3'-deoxythymidine (Bristol-Myers Squibb)

ddC

2',3'-dideoxycytidine (Roche)

ddI

2',3'-dideoxyinosine (Bristol-Myers Squibb)

DMP 266

a 1,4-dihydro-2H-3,1-benzoxazin-2-one

DMP 450

{[4R-(4-a,5-a,6-b,7-b)]-hexahydro-5,6-bis(hydroxy)-1,3-bis(3-amino)phenyl]methyl)-4,7-bis(phenylmethyl)-2{\it H}-1,3-diazepin-2-one}-bismesylate (Avid Therapeutics)

DP178

Synthetic peptide containing amino acids 127 to 162 of HIV-1 gp41

DXG

(-)-b-D-dioxolane-guanosine

EBU-dM

5-ethyl-1-ethoxymethyl-6-(3,5-dimethylbenzyl)uracil

E-EBU

5-ethyl-1-ethoxymethyl-6-benzyluracil

DS

dextran sulphate

E-EPSeU

1-(ethoxymethyl)-(6-phenylselenyl)-5-ethyluracil

E-EPU

1-(ethoxymethyl)-(6-phenyl-thio)-5-ethyluracil

F-ddA

2'-fluoro-2',3'-dideoxyadenosine

(-)-FTC

(-)-b-L-2',3'-dideoxy-5-fluoro-3'-thiacytidine (Triangle Pharmaceuticals)

HBY 097

(S)-4-isopropoxycarbonyl-6-methoxy-3-(methylthio-methyl)-3,4-dihydroquinoxalin-2(1H)-thione

HEPT

1-[(2-hydroxyethoxy)methyl]6-(phenylthio)thymine

JM2763

1,1'-(1,3-propanediyl)-bis-1,4,8,11-tetraazacyclo-tetradecane (Johnson Matthey)

JM3100

1,1'-[1,4-phenylenebis-(methylene)]bis-(1,4,8,11-tetraazacyclotetradecane) octahydrochloride dihydrate (Johnson Matthey)

KNI-272

(2S,3S)-3-amino-2-hydroxy-4-phenylbutyric acid-containing tripeptide

L-697,593

5-ethyl-6-methyl-3-(2-phthalimido-ethyl)pyridin-2(1H)-one

L-697,661

3-{[(-4,7-dichloro-1,3-benzoxazol-2-yl)methyl]amino}-5-ethyl-6-methylpyridin-2(1H)-one

L-FDDC

(-)-b-L-5-fluoro-2',3'-dideoxy-cytidine

L-FDOC

(-)-b-L-5-fluoro-dioxolane cytosine

MK-639

hydroxy-aminopentane amide HIV-1 protease inhibitor (Merck & Co)

MKC442

6-benzyl-1-ethoxymethyl-5-isopropyluracil (I-EBU, Triangle Pharmaceuticals/Mitsubishi)

MP-134

C2 symmetry-based protease inhibitor

MP-167

C2 symmetry-based protease inhibitor

nevirapine

11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyridol[3,2-b:2',3'-e] diazepin-6-one (Boehringer Ingelheim)

NNRTI

non-nucleoside reverse transcriptase inhibitor

NSC648400

1-benzyloxymethyl-5-ethyl-6-(alpha-pyridylthio)uracil (E-BPTU)

P9941

[2-pyridylacetyl-IIePheAla-y(CHOH)]\sub2 (Dupont Merck)

PFA

phosphonoformate (foscarnet, Astra)

PMEA

9-(2 phosphonylmethoxyethyl)adenine (Gilead Sciences)

PMPA

(R)-9-(2-phosphonyl-methoxypropyl)adenine (Gilead Sciences)

QM96521

A 1,1,3-trioxo-2H,4H-thieno[2,4-3][1,2,3]thiadiazine derivative (TTD)

Ro 31-8959

hydroxyethylamine derivative HIV-1 protease inhibitor (Roche)

RPI-312

1-[(3S)-3-(n-alpha-benzyloxycarbonyl)-l-asparginyl)-amino-2-hydroxy-4-phenyl-butyryl]-n-tert-butyl-l-proline amide (peptidyl protease inhibitor)

RPR103611

RT

reverse transcriptase

S-2720

6-chloro-3,3-dimethyl-4-(isopropenyl-oxycarbonyl)-3,4-dihydro-quinoxalin-2(1H)thione

SC-52151

hydroxyethylurea isostere protease inhibitor (Searle)

SC-55389A

hydroxyethyl-urea isostere protease inhibitor (Searle)

SDF-1a

Stromal cell-derived factor 1 a

TIBO R82150

(+)-(5S)-4,5,6,7-tetrahydro-5-methyl-6-(3-methyl-2-butenyl)-imidazo[4,5,1-jk][1,4]-benzodiazepin-2(1H)-thione (Janssen)

TIBO 82913

(+)-(5S)-4,5,6,7,-tetrahydro-9-chloro-5-methyl-6-(3-methyl-2-butenyl)-imidazo-[4,5,1-jk]-[1,4]benzo-diazepin-2(1H)-thione (Janssen)

TSAO-m3T

[2',5'-bis-O-(tert-butyl-dimethylsilyl)-3'-spiro-5'-(4'-amino-1',2'-oxathiole-2',2'-dioxide)]-b-D-pentofuranosyl-N3-methylthymine

U-90152

1-[3-[(1-methylethyl)-amino]-2-pyridinyl]-4-[[5-[(methylsulphonyl)-amino]-lH-indol-2yl]carbonyl]-piperazine

U-95133

(Alkylamino)piperidine bis(heteroaryl)piperizine analog

U-104489

(Alkylamino)piperidine bis(heteroaryl)piperizine analog

UC-040

thiocarboxanilide derivative (Uniroyal Chemical Co)

UC

thiocarboxanilide derivatives (Uniroyal Chemical Co)

UC-781

N-[4-chloro-3-(3-methyl-2-butenyloxy)phenyl]-2-methyl-3-furan-carbothioamide

UC-82

N-[4-chloro-3-(3-methyl-2-butenyloxy)phenyl]-2-methyl-3-thiophene-carbothioamide

VB 11,328

hydroxyethyl-sulphonamide protease inhibitor (Vertex Pharmaceuticals)

VX-478

hydroxyethylsulphonamide protease inhibitor (Vertex Pharmaceuticals)

XM 323

cyclic urea protease inhibitor (Dupont Merck)